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Biochemical Assay.
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Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to A1-adenosinereceptors in rat cerebral cortical membranes was assayed as described.
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Inhibition of binding by a range of concentrations of xanthine was assessed in triplicate in at least two separate experiments.
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Inhibition of 2-chloroadenosine-elicited  accumulation of [3H]cyclic  AMP accumulation in [3H]adenine-labeled guinea pig cerebral cortical slices was assayed as described in the presence of 10 pg/mL adenosine deaminase and 30 pM    4-[3-(cyclopentyloxy)-4-methoxyphenyl]-2-pyrrolidone (rolipram, ZK 62711).
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Inhibition of the response to 15 ¦ÌM 2-chloroadenosine by a range of concentrations of each xanthine was assessed in triplicate in at least two experiments. Ki values were calculated as described.
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