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Unless otherwise requested, primary screening in duplicate with quantitative data (e.g., IC50 ¡À SEM, Ki ¡À SEM and nH)
are shown where applicable for individual requested assays. In screening packages, primary screening in duplicate with
semi-quantitative data (e.g., estimated IC50, Ki and nH) are shown where applicable (concentration range of 4 log units);
available secondary functional assays are carried out (30 mM) and MEC or MIC determined only if active in primary assays
>50% at 1 log unit below initial test concentration.

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fjtony163: ½ð±Ò+10, ´ú·¢ 2016-03-16 18:06:18
fjtony163: ·­ÒëEPI+1, ´ú·¢ 2016-03-16 18:07:33
Unless otherwise requested, primary screening in duplicate with quantitative data (e.g., IC50 ¡À SEM, Ki ¡À SEM and nH) are shown where applicable for individual requested assays.
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In screening packages, primary screening in duplicate with
semi-quantitative data (e.g., estimated IC50, Ki and nH) are shown where applicable (concentration range of 4 log units);
ËùÓÐɸѡÖУ¬ÔÚÊʺϵÄŨ¶È·¶Î§£¬½áºÏ°ë¶¨Á¿Êý¾Ý(¼´Ëù¹À¼ÆµÄ IC50, Ki and nH)µÄ³õ²½µÄɸѡ£¨Ò»Ê½¶þ·Ý£©²Å»áÕ¹ÏÖ³ö¡£


available secondary functional assays are carried out (30 mM) and MEC or MIC determined only if active in primary assays >50% at 1 log unit below initial test concentration.
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2Â¥2016-01-29 21:47:03
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fjtony163: ½ð±Ò+10, ´ú·¢ 2016-03-16 18:06:26
³ýÁíÓÐÒªÇóÍ⣬³õɸ¶¨Á¿Öظ´Êý¾Ý£¨È磬IC50¡ÀSEM£¬Ki¡ÀSEMºÍNH£©¿ÉÓÃÓÚ¸öÀýÐèÇó²â¶¨¡£ÔÚɸ²é×é¼þÖУ¬³õɸ°ë¶¨Á¿Öظ´Êý¾Ý£¨È磬IC50Öµ/KiÖµºÍnHϵÊý´ÖÂÔÖµ£©¿ÉÓÃÓÚ£¨4¸ö¶ÔÊýµ¥Î»µÄŨ¶È·¶Î§ÄÚ£©Çé¿öϲⶨ; ½öµ±»îÐÔÔÚÒ»¼¶²â¶¨Å¨¶È>50£¥ÇÒµÍÓÚ³õʼÊÔÑéŨ¶È1¸ö¶ÔÊýµ¥Î»Ê±¿ÉÓÃÓÚ¶þ¼¶¹¦ÄÜ£¨30mM£©ºÍMEC»òMIC²â¶¨¡£

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nH= the Hill coefficientÏ£¶ûϵÊý£¨nH£©
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3Â¥2016-01-29 22:34:06
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liujie3214

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2Â¥: Originally posted by Î人һÐÄÒ»Òë at 2016-01-29 21:47:03
Unless otherwise requested, primary screening in duplicate with quantitative data (e.g., IC50 ¡À SEM, Ki ¡À SEM and nH) are shown where applicable for individual requested assays.
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3Â¥: Originally posted by sqlg888 at 2016-01-29 22:34:06
³ýÁíÓÐÒªÇóÍ⣬³õɸ¶¨Á¿Öظ´Êý¾Ý£¨È磬IC50¡ÀSEM£¬Ki¡ÀSEMºÍNH£©¿ÉÓÃÓÚ¸öÀýÐèÇó²â¶¨¡£ÔÚɸ²é×é¼þÖУ¬³õɸ°ë¶¨Á¿Öظ´Êý¾Ý£¨È磬IC50Öµ/KiÖµºÍnHϵÊý´ÖÂÔÖµ£©¿ÉÓÃÓÚ£¨4¸ö¶ÔÊýµ¥Î»µÄŨ¶È·¶Î§ÄÚ£©Çé¿öϲⶨ; ½öµ±»îÐÔÔÚ ...

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