±±¾©Ê¯ÓÍ»¯¹¤Ñ§Ôº2026ÄêÑо¿ÉúÕÐÉú½ÓÊÕµ÷¼Á¹«¸æ
²é¿´: 529  |  »Ø¸´: 3

781934544

гæ (³õÈëÎÄ̳)

[ÇóÖú] °ï·­ÒëÏÂÕâ¶Î£¬Ð»Ð»

This report describes the development and scale up of the synthesis of oxaisoxazolidinone 1, a significant synthon in the synthesis of the MRSA development compound AZD5847. Studies were carried out to ensure a short-term, risk based preparation of 9 on a 5 L scale with a solid isolation procedure and a safe, long-term manufacturing process for both 1 and 9 through extensive hazards evaluation.

·¢×ÔСľ³æIOS¿Í»§¶Ë

» ²ÂÄãϲ»¶

ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

781934544

гæ (³õÈëÎÄ̳)

2Â¥2016-01-11 13:21:59
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

781934544

гæ (³õÈëÎÄ̳)

3Â¥2016-01-12 08:39:53
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

ÂçÂçÒÀÈ»

°æÖ÷ (ÖªÃû×÷¼Ò)

ÓÅÐã°æÖ÷ÓÅÐã°æÖ÷ÓÅÐã°æÖ÷ÓÅÐã°æÖ÷ÓÅÐã°æÖ÷

¡¾´ð°¸¡¿Ó¦Öú»ØÌû

¡ï ¡ï ¡ï ¡ï ¡ï ¡ï ¡ï ¡ï ¡ï ¡ï
781934544: ½ð±Ò+10 2016-01-12 19:35:08
Õâ·Ý±¨¸æÃèÊöÁË·¢Õ¹·Å´óoxaisoxazolidinone 1µÄºÏ³É£¬ËüÊÇÒ»ÖÖÖØÒªµÄºÏ³ÉÏËάÔÚ ÓÉMRSAºÏ³É»¯ºÏÎï AZD5847¹ý³ÌÖС£Ñо¿±íÃ÷£¬ÎªÈ·±£¶ÌÆÚ·çÏÕ£¬9µÄÖÆ±¸ÔÚ5L¹ÌÌå·ÖÀë³ÌÐòÖнøÐС£¶ÔÓÚ1Óë9µÄ³¤ÆÚÖÆÔì¹ý³ÌӦͨ¹ý´óÁ¿Î£ÏÕÆÀ¹À¡£
¼È¿ÉÔç¾ÅÍíÎ壬Ҳ¿ÉÀ˼£ÌìÑÄ¡£
4Â¥2016-01-12 10:52:46
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû
Ïà¹Ø°æ¿éÌø×ª ÎÒÒª¶©ÔÄÂ¥Ö÷ 781934544 µÄÖ÷Ìâ¸üÐÂ
×î¾ßÈËÆøÈÈÌûÍÆ¼ö [²é¿´È«²¿] ×÷Õß »Ø/¿´ ×îºó·¢±í
[¿¼ÑÐ] Ò»Ö¾Ô¸ÎäÀí³µÁ¾×¨Ë¶×Ü·Ö 281 Çóµ÷¼Á +4 Éϰ¶Ñо¿Éú. 2026-04-02 4/200 2026-04-07 09:52 by ¼ÓÓÍÏòδÀ´°¡
[¿¼ÑÐ] 283·ÖÇóµ÷¼Á +11 ÊÔÊÔ¿´ß 2026-04-04 11/550 2026-04-07 09:52 by Öí»á·É
[¿¼ÑÐ] 304Çóµ÷¼Á +7 ËØÄê¼ÀÓï 2026-04-06 10/500 2026-04-06 23:31 by ËØÄê¼ÀÓï
[¿¼ÑÐ] ¹¤¿Æ 22408 267ÇóÍÆ¼ö +4 wanwan00 2026-04-05 5/250 2026-04-06 22:47 by chenzhimin
[¿¼ÑÐ] Ò»Ö¾Ô¸ÄϿƴóÉúÎïѧ297·Ö£¬Çóµ÷¼ÁÍÆ¼ö +6 Y-yyusx 2026-04-06 7/350 2026-04-06 22:39 by 52305043001
[¿¼ÑÐ] µ÷¼ÁÇóÖú£¨ÉúÎïÓëÒ½Ò©£© +3 @6952 2026-04-06 3/150 2026-04-06 21:48 by Ecowxq666£¡
[¿¼ÑÐ] 0703»¯Ñ§µ÷¼Á325·Ö +12 15771691647 2026-04-04 13/650 2026-04-06 12:00 by lijunpoly
[¿¼ÑÐ] ¿¼Ñе÷¼Á +5 ÃÀÀöµÄyouth_ 2026-04-04 6/300 2026-04-06 06:57 by houyaoxu
[¿¼ÑÐ] Ò»Ö¾Ô¸9²ÄÁÏѧ˶297ÒѹýÁù¼¶Çóµ÷¼ÁÍÆ¼ö +11 adaie 2026-04-04 12/600 2026-04-05 19:04 by À¶ÔÆË¼Óê
[¿¼ÑÐ] 298Çóµ÷¼Á +3 manman511 2026-04-05 3/150 2026-04-05 18:09 by kk112233
[¿¼ÑÐ] ¿¼Ñе÷¼Á +5 ËÄ´¨ÍõÌÎ 2026-04-04 5/250 2026-04-04 22:18 by à£à£à£0119
[¿¼ÑÐ] 333Çóµ÷¼Á +12 wfh030413@ 2026-04-03 13/650 2026-04-04 21:02 by jj987
[¿¼ÑÐ] 292Çóµ÷¼Á +11 2022080213 2026-04-04 13/650 2026-04-04 18:38 by macy2011
[¿¼ÑÐ] 291Çóµ÷¼Á +4 ÃÔÃÉľľ 2026-04-01 5/250 2026-04-04 15:59 by sihailian3
[¿¼ÑÐ] ±¾¿Æ211£¬×¨Òµ085404£¬293·ÖÇëÇóµ÷¼Á +5 Á«²Ë¾ÍÊÇź°É 2026-04-04 5/250 2026-04-04 14:08 by ÕâÊÇÒ»¸öÎÞÁĵÄê
[¿¼ÑÐ] ¿¼Ñе÷¼Á +8 ²»°®ºÈÒûÁÏ 2026-04-03 8/400 2026-04-03 16:40 by Mistake-J
[¿¼ÑÐ] 0805Çóµ÷¼Á +8 ÊÇË®·Ö 2026-03-31 8/400 2026-04-02 10:46 by guanxin1001
[¿¼ÑÐ] ¡¾Çóµ÷¼Á¡¿ÐÂÄÜÔ´²ÄÁϱ¾¿Æ£¬Ò»Ö¾Ô¸211£¬³õÊÔ321 +6 Çóµ÷¼ÁѧУ£¬ 2026-04-02 6/300 2026-04-02 09:41 by Çç¿Õ210210
[¿¼ÑÐ] 08¹¤¿Æ£¬295£¬½ÓÊÜ¿çרҵµ÷¼Á +6 lmnlzy 2026-03-31 6/300 2026-04-01 11:02 by ÄæË®³Ë·ç
[¿¼ÑÐ] Ò»Ö¾Ô¸Î÷µç085401ÊýÒ»Ó¢Ò»299Çóµ÷¼Á Áù¼¶521 +4 °®³Ô´óѼÀæ 2026-03-31 4/200 2026-03-31 11:51 by ²«»÷518
ÐÅÏ¢Ìáʾ
ÇëÌî´¦ÀíÒâ¼û