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781934544

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This report describes the development and scale up of the synthesis of oxaisoxazolidinone 1, a significant synthon in the synthesis of the MRSA development compound AZD5847. Studies were carried out to ensure a short-term, risk based preparation of 9 on a 5 L scale with a solid isolation procedure and a safe, long-term manufacturing process for both 1 and 9 through extensive hazards evaluation.

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781934544

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2楼2016-01-11 13:21:59
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781934544

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3楼2016-01-12 08:39:53
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781934544: 金币+10 2016-01-12 19:35:08
这份报告描述了发展放大oxaisoxazolidinone 1的合成,它是一种重要的合成纤维在 由MRSA合成化合物 AZD5847过程中。研究表明,为确保短期风险,9的制备在5L固体分离程序中进行。对于1与9的长期制造过程应通过大量危险评估。
既可早九晚五,也可浪迹天涯。
4楼2016-01-12 10:52:46
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