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十三

金虫 (正式写手)

[求助] 求稳定固体制剂辅料

非制剂专业,求相关知识,希望多多帮助

求稳定固体制剂辅料,保证化学药物制剂稳定

1:避免晶型转化

2、原料存在S和R构想,为S型入药,能保证构想稳定不转化的辅料都有哪些

求常规辅料,带构象辅料,特殊高分子材料,谢谢!
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jinkina

金虫 (正式写手)

【答案】应助回帖

★
十三(金币+1): 2011-06-14 08:11:00
qinhy(金币+1): 多谢回帖~~~ 2011-06-14 19:11:20
十三(金币+9): 2011-07-14 13:02:36
常用的就是MCC、淀粉、预胶化淀粉、乳糖、甘露醇等。
关于转不转晶,得通过实验才能确定,做晶型衍射
2楼2011-06-13 15:07:55
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