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Nat Prod Commun.  2016; 11(5):633-6 (ISSN: 1934-578X)
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609718476: ½ð±Ò+12, ¡ï¡ï¡ï¡ï¡ï×î¼Ñ´ð°¸ 2016-10-28 11:30:28
Silymarin versus Silibinin: Differential Antioxidant and Neuroprotective Effects against H2O2-induced Oxidative Stress in PC12 Cells
×÷Õß:Jiang, HH (Jiang, Hui-Hui)[ 1 ] ; Yan, FS (Yan, Fa-Shun)[ 1 ] ; Shen, L (Shen, Liang)[ 1 ] ; Ji, HF (Ji, Hong-Fang)[ 1 ]
NATURAL PRODUCT COMMUNICATIONS
¾í: 11  ÆÚ: 5  Ò³: 633-636
³ö°æÄê: MAY 2016
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The present study assessed comparatively the antioxidant activities of silymarin and its major active component silibinin and their neuroprotective effects against hydrogen peroxide (H2O2)-induced oxidative stress in rat pheochromocytoma PC12 cells. It was found that despite newly prepared silymarin and silibinin solution possessing comparable superoxide anion (O-2(center dot-))-scavenging activities, with time the activity of silymarin lowered slightly, but that of silibinin decreased dramatically. Both silymarin and silibinin suppressed H2O2 -induced oxidative stress and apoptosis, and the neuroprotective effect of silymarin was overall relatively stronger than that of silibinin. The findings provided clues for future studies on therapeutic potentials of the whole silymarin or purified silibinin for neurodegenerative diseases.
¹Ø¼ü´Ê
×÷Õ߹ؼü´Ê:Silymarin; Silibinin; Neurodegenerative diseases; Neuroprotective effects; PC12 cells
KeyWords Plus:THISTLE SILYBUM-MARIANUM; PARKINSONS-DISEASE; ALZHEIMERS-DISEASE; MILK THISTLE; NEURODEGENERATIVE DISEASES; MECHANISMS; MODEL; PREVALENCE; DISORDERS; APOPTOSIS
×÷ÕßÐÅÏ¢
ͨѶ×÷ÕßµØÖ·: Shen, L; Ji, HF (ͨѶ×÷Õß)
ÏÔʾÔöÇ¿×éÖ¯ÐÅÏ¢µÄÃû³Æ        Shandong Univ Technol, Sch Life Sci, Shandong Prov Res Ctr Bioinformat Engn & Tech, Zibo 255049, Peoples R China.
µØÖ·:
ÏÔʾÔöÇ¿×éÖ¯ÐÅÏ¢µÄÃû³Æ        [ 1 ] Shandong Univ Technol, Sch Life Sci, Shandong Prov Res Ctr Bioinformat Engn & Tech, Zibo 255049, Peoples R China
µç×ÓÓʼþµØÖ·:shen@sdut.edu.cn; jhf@sdut.edu.cn
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»ù½ð×ÊÖú»ú¹¹        ÊÚȨºÅ
Shandong Provincial Science Foundation for Distinguished Young Scholars        
JQ201508
Shandong Provincial Science Foundation        
ZR2015JL010
ZR2014CL008
²é¿´»ù½ð×ÊÖúÐÅÏ¢   
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NATURAL PRODUCTS INC, 7963 ANDERSON PARK LN, WESTERVILLE, OH 43081 USA
Àà±ð / ·ÖÀà
Ñо¿·½Ïòharmacology & Pharmacy; Food Science & Technology
Web of Science Àà±ð:Chemistry, Medicinal; Food Science & Technology
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ÎÄÏ×ÀàÐÍ:Article
ÓïÖÖ:English
Èë²ØºÅ: WOS:000375633500020
PubMed ID: 27319137
ISSN: 1934-578X
eISSN: 1555-9475
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Impact Factor (Ó°ÏìÒò×Ó): Journal Citation Reports®
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Web of Science ºËÐĺϼ¯ÖÐµÄ "±»ÒýƵ´Î": 0
3Â¥2016-10-28 11:14:58
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