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Intriguingly, the innovation of a fragment-based drug design (FBDD) approach has enabled rapid and efficient progress in drug discovery. In this critical review, we focus on the construction of fragment libraries and the advantages and disadvantages of various fragment-based screening (FBS) for constructing such libraries. We also highlight the deconstruction¨Creconstruction strategy by utilizing privileged fragments of reported ligands.

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2Â¥: Originally posted by 818james at 2016-01-10 22:32:38
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Intriguingly, the innovation of a fragment-based drug design (FBDD) approach has enabled rapid and efficient progress in drug discovery. In this critical review, we focus on the construction of fragment libraries and the advantages and disadvantages of various fragment-based screening (FBS) for constructing such libraries. We also highlight the¨Creconstruction strategy by utilizing privileged fragments of reported ligands.

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4Â¥: Originally posted by tonyhong1020 at 2016-01-12 11:17:27
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