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1?????ε??a????Y ??Υ?饶????10??mol/L???u??????133?N???ΙC??????????????塢????????????????????????Τ?????L?????????????????????M1??M2????M3?????塢????????5-HT2?????塢???????????弰??????????????????50????????躦????????????L?????????????????????M1????M3?????塢????????5-HT2????????????IC50????????????????????2.27??1.49??0.80????1.43??mol/L???????? 2????????a????Y ??1????????U??????????????????????Υ?饶???????c????Υ?饶??????0??30??100????600mg/kg?? ?g??U????????????????????Q?????????100mg/kg?????????????600mg/kg???????????????????仯??????6????1?????????????? ??2??????????????????? ??Υ?饶???????c????Υ?饶??????0.5??5????50??g/mL????hERG????躦???????????????0.5??g/mL??????????????hERG??????躦??????IC50????4.8??g/mL??????????o???E????????????R??????????????????????????????????餫?????????????????? ??3?????????????????? ???????????Υ?饶???????c????Υ?饶??????0??30??100????600mg/kg?? ?g??U???????κ??????????Q????????r?Q????????enhanced pause??Penh????????s?????????????????????600mg/kg?????4????8?r?g?????Q?????????r?Q?????ε????????8????4?????????????????????Τ???1????Penh?θ?????????????????????????v?S?????餫?????????? 4??????h????ΙC????I?C????????C??????¤??????Τ??????????????? 5 ?ыD??????路??????????Τ???D?????????????????Σ???????????ж?????????Τ????????????????Y???????????????????R????????40mg/???????????Υ?饶??????????AUC???μs28???????????????????????????P?????ε????????????????T???????β??????????K?????????????????????и???p?????i??????}????????????J?????????? 6 ?????Ф?D?????????????????????????????????????????????????????????????????Y?????????????Ф????Ф????????椵???????? |
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