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mary-juan

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[求助] 阿莫西林与他唑巴坦 已有1人参与

阿莫西林为什么不能与他唑巴坦类的联用?机制是什么?有相关文献吗
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guozhonglong

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【答案】应助回帖

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感谢参与,应助指数 +1
mary-juan: 金币+5, ★★★很有帮助, 5 2014-11-18 16:05:32
阿莫西林是β-内酰胺类抗生素,他唑巴坦是不可逆竞争型β-内酰胺酶抑制剂,通过抑制酶的活性,增加β-内酰胺类抗生素的抗菌活性,至于为什么二者不可连用,请参考以下这篇文献,希望对你有点帮助。
祝好~!

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