24小时热门版块排行榜    

查看: 714  |  回复: 3
当前只显示满足指定条件的回帖,点击这里查看本话题的所有回帖

liuxuekun

木虫 (小有名气)

[求助] 求助论文检索号,谢谢大侠!

Bai-Jun Ye, Xue-Kun Liu, Sheng-Ming Jiang, Xun Cui*, and Hu-Ri Piao*. Synthesis of 2-(4-Substitutedbenzyl-[1,4]diazepan-1-yl)-N-(1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolin-7-yl)acetamides as Inotropic Agents.
回复此楼

» 猜你喜欢

已阅   回复此楼   关注TA 给TA发消息 送TA红花 TA的回帖

baiyuefei

版主 (文学泰斗)

风雪

优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主优秀版主优秀版主

【答案】应助回帖

★ ★ ★
gruyclewee: 金币+3, 感谢应助,奖励一下。 2013-11-19 09:14:44
Synthesis of 2-(4-Substitutedbenzyl-[1,4]Diazepan-1-yl)-N-(1-Methyl-4,5-Dihydro-[1,2,4]Triazolo[4,3-A]Quinolin-7-Yl)Acetamides as Inotropic Agents  
作者: Ye, BJ (Ye, Bai-Jun)[ 2 ] ; Liu, XK (Liu, Xue-Kun)[ 2 ] ; Jiang, SM (Jiang, Sheng-Ming)[ 2 ] ; Cui, X (Cui, Xun)[ 1 ] ; Piao, HR (Piao, Hu-Ri)[ 2 ]  
来源出版物: CHEMICAL BIOLOGY & DRUG DESIGN  卷: 77   期: 1   页: 98-103   DOI: 10.1111/j.1747-0285.2010.01057.x   出版年: JAN 2011  
被引频次: 3 (来自 Web of Science)  
引用的参考文献: 10      [ 查看 Related Records ]     引证关系图引证关系图      
摘要: In an attempt to search for more potent positive inotropic agents, a series of N-(4,5-dihydro-1-methyl-[1,2,4]triazolo[4,3-a]quinolin-7-yl)-2-(substitutedbenzyl-[1,4]diazepan-1-yl)acetamides were synthesized and evaluated for positive inotropic activity by measuring left atrium stroke volume in isolated rabbit heart preparations. Some of these derivatives exhibited favorable activity compared with the standard drug, milrinone, among which 2-(4-(4-methylbenzyl)-[1,4]-diazepan-1-yl)-N-(4,5-dihydro-1-methyl-[1,2,4]triazolo[4,3-a]quinolin-7-yl)acetamide (6m) was the most potent, increasing stroke volume by 8.38 +/- 0.16% (milrinone 2.45 +/- 0.06%) at 3 x 10-5 m. The chronotropic effects of those compounds having inotropic effects were also evaluated in this work.  
入藏号: WOS:000285065000012  
文献类型: Article  
语种: English  
作者关键词: [1; 2; 4]triazolo[4; 3-a]quinolines; 1; 4-diazepan; positive inotropic activity; stroke volume  
KeyWords Plus: HEART-FAILURE; MORTALITY; VESNARINONE; ATRIA  
通讯作者地址: Cui, X (通讯作者) Yanbian Univ, Coll Preclin Med, Yanji 133000, Peoples R China.
  增强组织信息的名称
    Yanbian University  

地址:  [ 1 ] Yanbian Univ, Coll Preclin Med, Yanji 133000, Peoples R China
  增强组织信息的名称
    Yanbian University  
[ 2 ] Yanbian Univ, Coll Pharm, Minist Educ, Key Lab Nat Resources Changbai Mt & Funct Mol, Yanji 133000, Peoples R China
  增强组织信息的名称
    Yanbian University  

电子邮件地址: cuixun@ybu.edu.cn; piaohuri@yahoo.com.cn  
基金资助致谢:
基金资助机构 授权号
National Natural Science Foundation of China  30560177  

[显示基金资助信息][隐藏基金资助信息]   

This work was supported by the National Natural Science Foundation of China (No. 30560177).

出版商: WILEY-BLACKWELL PUBLISHING, INC, COMMERCE PLACE, 350 MAIN ST, MALDEN 02148, MA USA  
Web of Science 类别: Biochemistry & Molecular Biology; Chemistry, Medicinal  
研究方向: Biochemistry & Molecular Biology; Pharmacology & Pharmacy  
IDS 号: 691FF
3楼2013-11-17 19:41:47
已阅   回复此楼   关注TA 给TA发消息 送TA红花 TA的回帖
查看全部 4 个回答

baiyuefei

版主 (文学泰斗)

风雪

优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主优秀版主优秀版主

2楼2013-11-17 19:41:34
已阅   回复此楼   关注TA 给TA发消息 送TA红花 TA的回帖

baiyuefei

版主 (文学泰斗)

风雪

优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主文献杰出贡献优秀版主优秀版主优秀版主优秀版主优秀版主优秀版主

【答案】应助回帖

★ ★ ★ ★ ★ ★ ★ ★ ★ ★
liuxuekun: 金币+10, ★★★★★最佳答案 2013-12-17 08:30:09
WOS:000285065000012
4楼2013-11-17 19:42:16
已阅   回复此楼   关注TA 给TA发消息 送TA红花 TA的回帖
最具人气热帖推荐 [查看全部] 作者 回/看 最后发表
[考研] 一志愿北京化工大学材料与化工 264分各科过A区国家线 +3 哈哈157349 2026-03-21 3/150 2026-03-24 14:11 by zhyzzh
[考研] 资源与环境 调剂申请(333分) +6 holy J 2026-03-21 6/300 2026-03-24 09:51 by hengsmith
[考研] 一志愿武理材料工程348求调剂 +6  ̄^ ̄゜汗 2026-03-19 9/450 2026-03-23 19:53 by pswait
[考研] 考研化学308分求调剂 +7 你好明天你好 2026-03-23 8/400 2026-03-23 18:39 by macy2011
[考研] 一志愿中国石油大学(华东) 本科齐鲁工业大学 +4 石能伟 2026-03-17 4/200 2026-03-23 17:51 by 17862566385
[考研] 求调剂 +5 Zhangbod 2026-03-21 7/350 2026-03-22 13:13 by Zhangbod
[基金申请] 山东省面上项目限额评审 +4 石瑞0426 2026-03-19 4/200 2026-03-22 08:50 by Wei_ren
[考研] 085600材料与化工306 +4 z1z2z3879 2026-03-21 4/200 2026-03-21 23:44 by ms629
[考研] 材料与化工(0856)304求B区调剂 +3 邱gl 2026-03-20 7/350 2026-03-21 19:05 by 15709483992
[考研] 0703化学297求调剂 +3 Daisy☆ 2026-03-20 3/150 2026-03-21 17:45 by ColorlessPI
[考研] 279求调剂 +5 红衣隐官 2026-03-21 5/250 2026-03-21 14:59 by lature00
[考研] 22 350 本科985求调剂,求老登收留 +3 李轶男003 2026-03-20 3/150 2026-03-21 13:28 by 搏击518
[考研] 330求调剂0854 +3 assdll 2026-03-21 3/150 2026-03-21 13:01 by 搏击518
[考研] 304求调剂 +7 司空. 2026-03-18 7/350 2026-03-20 23:08 by JourneyLucky
[考研] 288求调剂 +16 于海海海海 2026-03-19 16/800 2026-03-20 22:28 by JourneyLucky
[考研] 求调剂,一志愿:南京航空航天大学大学 ,080500材料科学与工程学硕,总分289分 +4 @taotao 2026-03-19 4/200 2026-03-20 22:14 by JourneyLucky
[考研] 一志愿西南交通 专硕 材料355 本科双非 求调剂 +5 西南交通专材355 2026-03-19 5/250 2026-03-20 21:10 by JourneyLucky
[考研] 生物学调剂招人!!! +3 山海天岚 2026-03-17 4/200 2026-03-19 21:34 by 怎么释怀
[考研] 0703化学调剂 +4 18889395102 2026-03-18 4/200 2026-03-19 16:13 by 30660438
[考博] 26博士申请 +3 1042136743 2026-03-17 3/150 2026-03-17 23:30 by 轻松不少随
信息提示
请填处理意见