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cainiaodui

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There have been some notable clinical successes attributed to VEGF blockade, and Avastin is approved for treatment of colon and renal cancers; however, many cancers that clearly require vascularization are highly resistant to VEGF-A blockade from the start. In addition, many others acquire such resistance, casting some doubt both on the therapeutic benefit of VEGF-A blockade and on the factor’s indispensability in angiogenesis. Drug developers have more recently sought to target other known angiogenic pathways, pursuing therapies that might be useful independently or in concert with VEGF blockade in the treatment of cancer.
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xux730

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cainiaodui: 金币+5, 翻译EPI+1 2013-09-26 18:56:36
已经有一些显著的、归因于阻滞血管内皮生长因子的成功的临床案例,如Avastin已被批准用于治疗结肠癌和肾癌;但是,许多明确需要新血管生成支撑的癌症从一开始就具有很强的针对VEGF-A阻断剂的耐受性。此外,其它许多种癌症也获得这种耐受性,这些对VEGF-A阻断剂及对血管生成不可少的因子对癌症治疗的益处投下阴影。药物开发商最近试图针对其他已知的血管生成途径,追求独立于VEGF-A阻断剂或与VEGF-A阻断剂协同的、有用的癌症治疗方法。
2楼2013-09-23 12:37:45
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