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Incubations from previously frozen, matching pooled human liver S-9 and cytosol from 10 donors contained 1 mg/ml cytosol or 2.5 mg/ml S-9 fraction in 100 mM potassium phosphate buffer (pH 7.4) and initiated with substrate [(1 ¦ÌM) final organic vehicle concentration was 0.01% dimethyl sulfoxide and 0.6% acetonitrile], with a final reaction volume of 200 ¦Ìl.

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