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The authors use concentration units of ug/ml throughout the manuscript and in the figures. It is more customary to use molarity-based units (nM, uM, mM, etc.) when presenting biological characterization of "small molecule" therapeutics (as opposed to biological therapeutics such as antibodies, etc.).  The authors are strongly encouraged to change all concentration units to molarity-based units, throughout the manuscript and in the figures (the exception would be doses used in vivo studies, which should be presented in mg/kg units).
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