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Adipocytes differentiate from preadipocytes.  Transcription factors including PPAR¦Ã (peroxisome proliferator-activated receptor ¦Ã), C/EBP family (CCAAT/enhancer binding proteins; C/EBR¦Á, C/EBR¦Â and C/EBR¦Ä) and ADD1/SREBP1c (adipocyte determination differentiation factor 1)/(sterol regulatory element binding protein 1c) play a crucial role in adipocyte differentiation.  The expression of these transcription factors is induced at different points of time in the course of adipocyte differentiation and they interact with one another to regulate adipocyte-specific genes and progressively induce fat metabolism and adipocyte differentiation .
Accordingly, a material that has the activity of regulating differentiation from preadipocytes to adipocytes and/or fat accumulation in adipose tissues or suppressing the expression of PPAR¦Ã, C/EBR¦Á, and/or ADD1/SREBP1c may be used as an anti-obesity agent.  As such, ginkgolide A or bilobalide isdisclosed in Korean Patent No. 920648, ginsenoside-Rf or compound K in Korean Patent No. 847252, and oltipraz inKorean Patent No. 576157.
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