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As no development has been reported for some time, this program is assumed to be discontinued. Pfizer (formerly by Warner-Lambert), under license from the University of Auckland, was developing canertinib (CI-1033, PD-0183805), a water soluble, orally-available analog of PD-169414, an EGFR tyrosine kinase inhibitor, as a potential treatment for cancer [427113]. By January 2000, phase I trials were underway [353284], [352930]. In September 2001, the drug was reported to be in phase II trials [427113], [429152]; these trials were ongoing in June 2004 [542422]. |
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