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右岸

金虫 (正式写手)

[求助] canertinib卡奈替尼这个抗肿瘤药物有没有上市?

canertinib卡奈替尼这个抗肿瘤药物有没有上市?如果有,什么时候?
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hongju

捐助贵宾 (小有名气)

【答案】应助回帖

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zhoudeli(金币+1): 多谢参与。 2011-12-25 17:47:35
mouse103: 应助指数+1 2012-05-20 05:30:39
右岸: 金币+2, 有帮助 2012-06-01 22:12:38
As no development has been reported for some time, this program is assumed to be discontinued.

Pfizer (formerly by Warner-Lambert), under license from the University of Auckland, was developing canertinib (CI-1033, PD-0183805), a water soluble, orally-available analog of PD-169414, an EGFR tyrosine kinase inhibitor, as a potential treatment for cancer [427113]. By January 2000, phase I trials were underway [353284], [352930]. In September 2001, the drug was reported to be in phase II trials [427113], [429152]; these trials were ongoing in June 2004 [542422].

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2楼2011-12-25 16:13:43
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右岸

金虫 (正式写手)

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: Originally posted by hongju at 2011-12-25 16:13:43:
As no development has been reported for some time, this program is assumed to be discontinued.

Pfizer (formerly by Warner-Lambert), under license from the University of Auckland, was developing  ...

谢谢
3楼2011-12-25 17:27:13
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ashuai078201

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感谢参与,应助指数 +1
mouse103: 金币+1, 谢谢参与 2012-05-20 05:31:16
由于没有发展已经报道了一段时间,这个方案是假设终止。
给翻译下
4楼2011-12-27 15:10:41
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chem_gd

金虫 (初入文坛)

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感谢参与,应助指数 +1
mouse103: 金币+1, 谢谢参与 2012-05-20 05:31:33
没有上市。辉瑞还有后续的类似分子,以及Boehringer Ingelheim也有类似分子,但是效果不是很好。
5楼2012-04-02 11:11:18
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