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This critical review focuses on the anti-cancer fight using gold nanoparticles (AuNPs)functionalized with chemotherapeutic drugs in so-called ¡®¡®complexes¡¯¡¯ (supramolecular assemblies)and ¡®¡®conjugates¡¯¡¯ (covalent assemblies) as vectors. There is a considerable body of recentliterature on various tumor-imaging techniques using the surface plasmon band (SPB) and the¡®¡®passive¡¯¡¯ and ¡®¡®active¡¯¡¯ vectorization of anti-cancer drugs. This article reviews the main conceptsand the most recent literature data with emphasis on AuNP preparation,cytotoxicities and usein selective targeting of cancer cells with over-expressed receptors for diagnosis and therapy
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