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qiuyuekaixin

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Candesartan-celexetil was first dissolved as a 1-mg/ml stock solution
in polyethylene glycol 400/ethanol/Cremophor EL (Sigma)/water (10/5/2/83%), adjusted to pH 9 with 0.2 M Na2CO3.The solution was diluted in water to a final concentration equal to or less than 1/0.5/0.2% PEG/ethanol/Cremophor EL.

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zhaochenchuo

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qiuyuekaixin(½ð±Ò+8, ·­ÒëEPI+1): лл£¡ 2011-05-13 17:29:00
Ê×ÏȽ«¿²µØÉ³Ì¹Î÷õ¥ÈÜÓÚPEG400-ÒÒ´¼-¾ÛÑõÒÒÏ©±ÍÂéÓÍ£¨sigma£©-Ë®£¨10:5:2:83£©ÈÜÒºÖУ¬ÖƳÉ1mg/ml´¢±¸Òº£¬ÓÃ0.2mol/l Na2CO3µ÷pHÖÁ9¡£½«´ËÈÜÒºÓÃˮϡÊÍÖÁÖÕŨ¶ÈµÈÓÚ»òµÍÓÚ1/0.5/0.2%PEG/ÒÒ´¼/¾ÛÑõÒÒÏ©±ÍÂéÓÍ¡£
2Â¥2011-05-13 17:19:18
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yinjuanchen

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Originally posted by qiuyuekaixin at 2011-05-13 16:53:21:
Candesartan-celexetil was first dissolved as a 1-mg/ml stock solution
in polyethylene glycol 400/ethanol/Cremophor EL (Sigma)/water (10/5/2/83%), adjusted to pH 9 with 0.2 M Na2CO3.The solution wa ...

µÚÒ»¸öµ¥´Ê¾Í·­²»ºÃ£¬ÕûÌåÉÏÊÇÓþÛÒÒ¶þ´¼400Åä³É1mg/mlµÄÔ­ÈÜÒº£¬ÆäÖÐÒÒÃÑ/¿ËÁÐĪ·ðEL/Ë®µÄÖÊÁ¿·ÖÊýΪ(10/5/2/83%),È»ºóÓÃ0.2M̼ËáÄÆÈÜÒºµ÷½ÚPHµ½9£¬ÈÜÒº×îºóÓÃË®ÕôÁóʹÉÏÊöÿÖÖÎïÖʵÄÖÊÁ¿·ÖÊý²»´óÓÚ1//0.5/0.2%.
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3Â¥2011-05-13 17:20:05
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yinjuanchen

Ìú¸Ëľ³æ (ÖøÃûдÊÖ)

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Originally posted by yinjuanchen at 2011-05-13 17:20:05:
µÚÒ»¸öµ¥´Ê¾Í·­²»ºÃ£¬ÕûÌåÉÏÊÇÓþÛÒÒ¶þ´¼400Åä³É1mg/mlµÄÔ­ÈÜÒº£¬ÆäÖÐÒÒÃÑ/¿ËÁÐĪ·ðEL/Ë®µÄÖÊÁ¿·ÖÊýΪ(10/5/2/83%),È»ºóÓÃ0.2M̼ËáÄÆÈÜÒºµ÷½ÚPHµ½9£¬ÈÜÒº×îºóÓÃË®ÕôÁóʹÉÏÊöÿÖÖÎïÖʵÄÖÊÁ¿·ÖÊý²»´óÓÚ1//0.5/0.2%.

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4Â¥2011-05-13 17:23:28
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qiuyuekaixin

гæ (СÓÐÃûÆø)

ÒýÓûØÌû:
Originally posted by zhaochenchuo at 2011-05-13 17:19:18:
Ê×ÏȽ«¿²µØÉ³Ì¹Î÷õ¥ÈÜÓÚPEG400-ÒÒ´¼-¾ÛÑõÒÒÏ©±ÍÂéÓÍ£¨sigma£©-Ë®£¨10:5:2:83£©ÈÜÒºÖУ¬ÖƳÉ1mg/ml´¢±¸Òº£¬ÓÃ0.2mol/l Na2CO3µ÷pHÖÁ9¡£½«´ËÈÜÒºÓÃˮϡÊÍÖÁÖÕŨ¶ÈµÈÓÚ»òµÍÓÚ1/0.5/0.2%PEG/ÒÒ´¼/¾ÛÑõÒÒÏ©±ÍÂéÓÍ¡£

Groups of six animals received oral candesartan-cilexetil (TCV-116; ASTRA,Mo ¡§ lndal, Sweden) at 10mg/kg per day for 14 days or received vehicle, both dissolved in their drinking water. Candesartan-cilexetil was first dissolved as a 1 mg/ml stock solution in polyethylene glycol400/ethanol/Cremophor EL (Sigma)/water (10/5/2/83%), adjusted to pH 9 with 0.2 M Na2CO3. The solution was diluted in water to a final concentration 1/0.5/0.2 polyethylene
glycol 400/ethanol/Cremophor EL.
Õâ¶ÎºÍÄǶÎÖ÷ÒªÒâ˼ÊÇÒ»ÑùµÄ£¬Èç¹ûÓÐʱ¼ä°ïÎÒ·­Ò»ÏÂÕâ¶Î£¡·Ç³£¸Ðл£¡
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5Â¥2011-05-13 17:32:21
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zhaochenchuo

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qiuyuekaixin(½ð±Ò+2): ·Ç³£¸Ðл£¡ 2011-05-13 18:23:40
6×鶯Îï¿Ú·þ¸øÓ迲µØÉ³Ì¹Î÷õ¥£¨TCV-116; ASTRA,Mo ¡§ lndal, Sweden£©»ò¸¨ÁÏ£¬¾ùÈÜÓÚÆäÒûÓÃË®ÖиøÒ©£¬Ã¿Ìì10mg/kg£¬¸øÒ©14Ìì¡£
6Â¥2011-05-13 17:41:04
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qiuyuekaixin

гæ (СÓÐÃûÆø)

ÒýÓûØÌû:
Originally posted by zhaochenchuo at 2011-05-13 17:41:04:
6×鶯Îï¿Ú·þ¸øÓ迲µØÉ³Ì¹Î÷õ¥£¨TCV-116; ASTRA,Mo ¡§ lndal, Sweden£©»ò¸¨ÁÏ£¬¾ùÈÜÓÚÆäÒûÓÃË®ÖиøÒ©£¬Ã¿Ìì10mg/kg£¬¸øÒ©14Ìì¡£

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7Â¥2011-05-13 18:24:46
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