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A l¡¯instar du mod¨¨le animal, chez l¡¯homme, le pirib¨¦dil se m¨¦tabolise en trois m¨¦tabolites principaux, un d¨¦riv¨¦ hydroxyl¨¦, un d¨¦riv¨¦ dihydroxyl¨¦ et un d¨¦riv¨¦ trihydroxyl¨¦, qui sont tous ¨¦limin¨¦s essentiellement par voie urinaire.Apr¨¨s administration orale r¨¦p¨¦t¨¦e du pirib¨¦dil chez des patients parkinsoniens, la demi-vie d¡¯¨¦limination moyenne de la mol¨¦cule m¨¨re est d¡¯environ 20 heures.
Ces donn¨¦es justifient l¡¯utilisation de cette mol¨¦cule en trois doses quotidiennes chez les patients parkinsoniens et afin d¡¯¨¦viter la pr¨¦sence de pics de concentration pendant la journ¨¦e ¨¤ l¡¯¨¦tat d¡¯¨¦quilibre.

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