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Benzothiazole derivative are known as inhibitors of
topoisomerase II, tyrosine kinase, Clk 1/4, ubiquitin proteasome
system and mitochondrial respiration [13¨C16]. It has
been reported that benzothiazoles potently block glutamate
neurotransmission both at presynaptic and postsynaptic
levels, inhibit huntingtin aggregation in cell culture,
increase intracellular Ca2+ [6]. Some benzothiazoles induce
cell cycle arrest, activate caspases, target CYP1 and interact
with DNA molecule
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Originally posted by ÎÞè¦ at 2009-10-29 11:33:
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