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Bioorganic & Medicinal Chemistry Letters
Volume 24, Issue 16, 15 August 2014, Pages 3869¨C3876

¡¾2¡¿Discovery of potent and selective urea-based ROCK inhibitors: Exploring the inhibitor¡¯s potency and ROCK2/PKA selectivity by 3D-QSAR, molecular docking and molecular dynamics simulations
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ͨѶ×÷ÕßµØÖ·: Cheng, LP (ͨѶ×÷Õß)
Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China.
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[ 1 ] Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China
[ 2 ] E China Univ Sci & Technol, Sch Chem & Mol Engn, Key Lab Adv Mat, Shanghai 200237, Peoples R China
[ 3 ] E China Univ Sci & Technol, Sch Chem & Mol Engn, Inst Fine Chem, Shanghai 200237, Peoples R China
µç×ÓÓʼþµØÖ·:chengliping@sit.edu.cn
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National Natural Science Foundation of China  
21172148
Scientific Research Innovation Project of Shanghai  
14YZ148
'College Students' Innovative Activities' of Shanghai  
PE2014044
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PERGAMON-ELSEVIER SCIENCE LTD, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD OX5 1GB, ENGLAND
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Ñо¿·½Ïòharmacology & Pharmacy; Chemistry
Web of Science Àà±ð:Chemistry, Medicinal; Chemistry, Organic
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ÎÄÏ×ÀàÐÍ:Article
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Èë²ØºÅ: WOS:000340565900038
PubMed ID: 25022881
ISSN: 0960-894X
eISSN: 1464-3405
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Web of Science ºËÐĺϼ¯ÖÐµÄ "ÒýÓõIJο¼ÎÄÏ×": 33
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Shanghai Inst Technol, Sch Chem & Environm Engn, 100 Hai Quan Rd, Shanghai 201418, Peoples R China.
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[ 1 ] Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China
[ 2 ] Chinese Acad Sci, Shanghai Inst Organ Chem, Key Lab Synthet Chem Nat Subst, Shanghai 200032, Peoples R China
[ 3 ] Scripps Res Inst, Med Chem, Translat Res Inst, Jupiter, FL 33458 USA
µç×ÓÓʼþµØÖ·:yinyan@sit.edu.cn; yfeng@scripps.edu
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Science and Technology Commission of Shanghai Municipality  
12ZR1431100
National Natural Science Foundation of China  
21172148
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PERGAMON-ELSEVIER SCIENCE LTD, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD OX5 1GB, ENGLAND
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Ñо¿·½Ïò:Biochemistry & Molecular Biology; Pharmacology & Pharmacy; Chemistry
Web of Science Àà±ð:Biochemistry & Molecular Biology; Chemistry, Medicinal; Chemistry, Organic
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ÎÄÏ×ÀàÐÍ:Article
ÓïÖÖ:English
Èë²ØºÅ: WOS:000353380400020
PubMed ID: 25882521
ISSN: 0968-0896
eISSN: 1464-3391
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IDS ºÅ: CG6BM
Web of Science ºËÐĺϼ¯ÖÐµÄ "ÒýÓõIJο¼ÎÄÏ×": 35
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