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taozhu006: ½ð±Ò+30, ¡ï¡ï¡ï¡ï¡ï×î¼Ñ´ð°¸ 2015-06-25 17:49:46
Synthesis of Main Impurity of Vildagliptin

×÷Õß:Tao, Z (Tao, Zhu)[ 1 ] ; Deng, Y (Deng, Yu)[ 1 ] ; Chen, YJ (Chen, Yingjie)[ 1 ] ; Wang, AM (Wang, Anmin)[ 1 ] ; Hu, XN (Hu, Xiangnan)[ 1 ]

ASIAN JOURNAL OF CHEMISTRY

¾í: 26

ÆÚ: 12

Ò³: 3489-3492

×Ó¼­: B

³ö°æÄê: JUN 2014

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A four-step synthesis of the main impurity of vildagliptin has been easily accomplished with high-yielding starting from L-proline. This compound can be used as a reference marker in an analytical method to determine the chemical purity of the vildagliptin.
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×÷Õ߹ؼü´ÊPP-IV inhibitors; Vildagliptin; L-proline; Impurity

KeyWords Plus:TYPE-2 DIABETES-MELLITUS; DIPEPTIDYL PEPTIDASE-4 INHIBITOR; SAXAGLIPTIN; SITAGLIPTIN; ALOGLIPTIN; THERAPY
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ͨѶ×÷ÕßµØÖ·: Hu, XN (ͨѶ×÷Õß)
[ÏÔʾÔöÇ¿×éÖ¯ÐÅÏ¢µÄÃû³Æ]         Chongqing Med Univ, Coll Pharmaceut Sci, Chongqing 400016, Peoples R China.

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[ÏÔʾÔöÇ¿×éÖ¯ÐÅÏ¢µÄÃû³Æ]         [ 1 ] Chongqing Med Univ, Coll Pharmaceut Sci, Chongqing 400016, Peoples R China

µç×ÓÓʼþµØÖ·:huxiangnan62@163.com
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Natural Science Foundation of Chongqing (CSTC)        
2006BB5286
Chongqing Medical University          
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ASIAN JOURNAL OF CHEMISTRY, 11/100 RAJENDRA NAGAR, SECTOR 3,, SAHIBABAD 201 005, GHAZIABAD, INDIA
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Ñо¿·½Ïò:Chemistry

Web of Science Àà±ð:Chemistry, Multidisciplinary
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ÎÄÏ×ÀàÐÍ:Article

ÓïÖÖ:English

Èë²ØºÅ: WOS:000343762400011

ISSN: 0970-7077

eISSN: 0975-427X
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    Impact Factor (Ó°ÏìÒò×Ó): Journal Citation Reports®

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Web of Science ºËÐĺϼ¯ÖÐµÄ "ÒýÓõIJο¼ÎÄÏ×": 23

Web of Science ºËÐĺϼ¯ÖÐµÄ "±»ÒýƵ´Î": 0
2Â¥2015-06-25 17:46:31
ÒÑÔÄ   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

youyouyanr

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Cloning and Characterization of Glyceraldehyde-3-Phosphate Dehydrogenase from Orchid (Cymbidium goeringii)  

저자: Tian, Yun-Fang; Li, Han; Yuan, Xiu-Yun; 등등.

ASIAN JOURNAL OF CHEMISTRY  권: 26   호: 17   페이지: 5321-5323   부: A   출판연도: SEP 2014

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