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The relationship between autophagy and apoptosis is very
complex, and the signalling pathways of autophagy and apoptosis
are extensively interconnected. 17 The ability of Ir-2 to induce
apoptosis in A549 cells was investigated by an annexin V staining
assay measured by flow cytometry (Fig. S10a, ESI† and confocal
microscopy (Fig. S10b, ESI†. Compared with the vehicle-treated
control cells (5.1 ? 0.5%), only negligible fractions of the A549 cells
became annexin V-positive after treatment with Ir-2 (2 mM: 6.3 ?
0.7%; 4 mM: 8.5 ? 1.0%). However, a considerable percentage of
cells underwent apoptosis upon cisplatin treatment (25 mM: 34.3 ?
2.9%; 50 mM: 48.6 ? 4.2%)
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