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ÊéÃû A Pharmacology Primer, Theory, Applications, and Methods
×÷ÕßTerry Kenakin
Ò³Êý 294
³ö°æÉçAcademic Press
ISBN 9780123705990
Ŀ¼1.1 ABOUT THIS BOOK 1
1.2 WHAT IS PHARMACOLOGY? 1
1.3 THE RECEPTOR CONCEPT 2
1.4 PHARMACOLOGICAL TEST SYSTEMS 4
1.5 THE NATURE OF DRUG RECEPTORS 6
1.6 PHARMACOLOGICAL INTERVENTION
AND THE THERAPEUTIC
LANDSCAPE 6
1.7 SYSTEM-INDEPENDENT DRUG
PARAMETERS: AFFINITY AND
EFFICACY 9
1.8 WHAT IS AFFINITY? 10
1.9 THE LANGMUIR ADSORPTION
ISOTHERM 10
1.10 WHAT IS EFFICACY? 13
1.11 DOSE-RESPONSE CURVES 14
1.12 CHAPTER SUMMARY AND
CONCLUSIONS 18
1.13 DERIVATIONS: CONFORMATIONAL
SELECTIONS AS A MECHANISM OF
EFFICACY 18
References 19¡ï¡ï¡ï¡ï¡ï¡ï¡ï2014Êé¼®³¬¼¶ÌûÈýÆßÁù¡¶Ò©ÀíѧÈëÃÅ£¬ÀíÂÛ£¬Ó¦Ó㬷½·¨¡·
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