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A number of investigations have been conducted in the past two decades to improve the understanding of the therapeutic prospects of GST. The involvement of GST in drug resistances has created an alternative target in the enhancement of potency of therapeutic agents. A rationale has been established to utilize agents that selectively inhibit the various classes of GST as adjuvant in anticancer chemo- therapy and as antiparasitic drugs. This concept was formu- lated in a bid to discover compounds that can inactivate GST for enhanced activity of the desired drug. These agents could act by either inhibiting the catalytic activity of GST in metabolism of electrophilic drugs [28] or in disruption of the complex formed between GST and stress signal kinases ¡£ |
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RXMCDM: ½ð±Ò+1, ¶àлӦÖú£¡ 2014-03-10 13:00:47
wzg389960: ½ð±Ò+20, ·ÒëEPI+1, ¡ï¡ï¡ï¡ï¡ï×î¼Ñ´ð°¸ 2014-03-10 13:34:32
RXMCDM: ½ð±Ò+1, ¶àлӦÖú£¡ 2014-03-10 13:00:47
wzg389960: ½ð±Ò+20, ·ÒëEPI+1, ¡ï¡ï¡ï¡ï¡ï×î¼Ñ´ð°¸ 2014-03-10 13:34:32
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2Â¥2014-03-10 12:59:32
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- ×¢²á: 2011-10-22
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3Â¥2014-03-10 13:35:38
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- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 1023.7
- Ìû×Ó: 157
- ÔÚÏß: 39.4Сʱ
- ³æºÅ: 1455748
- ×¢²á: 2011-10-22
- ÐÔ±ð: GG
- רҵ: ÌìÈ»Óлú»¯Ñ§

4Â¥2014-03-10 14:59:12














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