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yin198716

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What about the ways of DLL4 targeting? As mentioned above, one of them is specific targeting using anti-DLL4 antibodies. Unlike γ-secretase inhibitors, anti-DLL4 antibodies did not induce gastrointestinal toxicity. They have no discernible impact on goblet cell differentiation or crypt progenitor cell proliferation. Hoey et al. found that selective antihuman antibody 21M18 inhibited expression of Notch target genes including HES1 and ATOH1, which in effect caused a low level of malignant cell proliferation .
Oncology
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RXMCDM

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yin198716: 金币+5, 翻译EPI+1 2014-02-24 15:34:00
DLL4靶向方式是怎么样的?如上所述,其中之一是特定的抗DLL4抗体靶向。与γ-分泌酶抑制因子不同,抗DLL4抗体不诱导胃肠道毒性。他们对杯状细胞分化或隐窝祖细胞的增殖没有明显的影响。Hoey等发现抗人抗体21M18选择性抑制包括HES1基因和ATOH1基因在内的Notch靶基因,抑制靶基因实际上造成了恶性细胞增殖水平低下。
供参考!
?
2楼2014-02-22 01:18:42
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3楼2014-02-23 16:01:53
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