±±¾©Ê¯ÓÍ»¯¹¤Ñ§Ôº2026ÄêÑо¿ÉúÕÐÉú½ÓÊÕµ÷¼Á¹«¸æ
²é¿´: 1676  |  »Ø¸´: 6
µ±Ç°Ö»ÏÔʾÂú×ãÖ¸¶¨Ìõ¼þµÄ»ØÌû£¬µã»÷ÕâÀï²é¿´±¾»°ÌâµÄËùÓлØÌû

mollyzhang

Ìú¸Ëľ³æ (ÖøÃûдÊÖ)

[ÇóÖú] ÇóÖú¹ØÓÚרÀû²éѯµÄÒ»¸öÎÊÌâ!

×î½ü×÷¹ØÓÚÒ»¸ö°ÐµãµÄÎÄÏ×µ÷ÑÐ,
²éÁ˼¸¼Ò¹«Ë¾£¬
ÈçPamlico Pharmaceutical Inc£¬Axxam£¬Advinus Therapeutics,ÔÚÆä¹«Ë¾Ö÷Ò³ÉÏÓйØÓÚGPR120µÄÐÅÏ¢,µ«ÊÇÎÞÂÛ²éscifinder,»¹ÊÇderwent£¬»¹ÊÇÔÚÅ·ÖÞרÀû¾ÖºÍÃÀ¹úרÀû¾Ö¶¼Ã»ÓÐÕÒµ½¸Ã¹«Ë¾¸Ã°ÐµãµÄרÀû¡£ÏëÇë½Ìר¼ÒÊÇûÓÐÉêÇëרÀû£¿»¹ÊÇûÓй«¿ª£¿¡¡
ÔÚÌÀÄ·Ñ·Öв鵽µÄÐÅÏ¢
Pamlico Pharmaceutical is investigating    a G-protein coupled receptor 120  (GPR120) agonist for the potential treatment of  diabetes. In September 2011, the program was in lead optimization  [1226961]; in March 2013, this was still the case  [1390000]. In September 2011,  the company was seeking to outlicense its programs [1226961].
ÔÚ£²£°£±£±Äê¸Ã¹«Ë¾¾ÍÔÚoutlicense its programs£¬ÄÇÓ¦¸ÃÓÐרÀûÁ˰ɣ¿¡¡ÎªÊ²Ã´²é²»µ½ÄØ£¿

¸Ã¹«Ë¾ÍøÕ¾
http://www.pamlicopharma.com/Home/research


»¹ÓÐAxxam¡¡
http://www.axxam.com/discoverypro/discpro.asp

Advinus Therapeutics
http://www.advinus.com/pipeline.asp
ÔÚÌÀÄ·Ñ·Öв鵽µÄÐÅÏ¢
Advinus Therapeutics is investigating dual agonists of GPR40 and GPR120, for the potential treatment of type 2 diabetes [1231883], [1488118]. In October 2011, the program was in discovery and target identification was underway [1231883]; in October 2013, the program was listed as being under hit-to-lead development [1488118].   In October 2011, the company was seeking to outlicense the programs [1231883].

ÒÔÉϼ¸¼Ò¹«Ë¾¶¼²é²»µ½Æä¸Ã°ÐµãµÄרÀû£¬Çóר¼Ò½â»ó£¡²»Ê¤¸Ð¼¤£¡
»Ø¸´´ËÂ¥

» ²ÂÄãϲ»¶

» ±¾Ö÷ÌâÏà¹Ø¼ÛÖµÌùÍÆ¼ö£¬¶ÔÄúͬÑùÓаïÖú:

ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

whatt

ľ³æ (ÕýʽдÊÖ)

¡¾´ð°¸¡¿Ó¦Öú»ØÌû

¡ï ¡ï ¡ï ¡ï ¡ï
mollyzhang: ½ð±Ò+40 2013-11-12 09:42:02
yuanahen: ½ð±Ò-29, Â¥Ö÷·´À¡²Ù×÷ʧÎóʵ¼ÊÊÇ+5·Ö 2013-11-12 13:49:20
yuanahen: ½ð±Ò-6, Â¥Ö÷·´À¡´íÎó 2013-11-12 13:49:51
ÒýÓûØÌû:
4Â¥: Originally posted by mollyzhang at 2013-11-11 15:37:04
ÎÒÊÇÒòΪÔÚÌÀÄ·Ñ·Öв鵽ÒÔÉϵĹ«Ë¾ÔÚ×ö¸Ã°Ðµã, ËùÒÔÊÇÒÔ¹«Ë¾Ãû³Æ¼ìË÷µÄ,Æä´ÎÎÒÒÔ GPR120 (FFA4)Ò²¶¼Ã»ËÑË÷µ½ÉÏÊö¹«Ë¾µÄרÀû...

ÎÒÒ²¾­³£×öרÀûÎÄÏ׵ļìË÷£¬ÓÐʱºòÐèҪͨ¹ý¶àÖÖ;¾¶²ÅÄÜÃüÖÐÄ¿±ê¡£½¨ÒéÓÃÏà¹ØÊÊӦ֢Ϊ¼ìË÷´Ê£¬È»ºóÔÙÖð²½ÒÔ¹«Ë¾Ãû³Æ¡¢°ÐµãÃû³ÆµÈËõС·¶Î§¡£

[ ·¢×ÔСľ³æ¿Í»§¶Ë ]
ÐÄÓжà´ó£¬Ìì¿Õ¾ÍÓжà´ó£¡£¡
7Â¥2013-11-11 22:12:55
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû
²é¿´È«²¿ 7 ¸ö»Ø´ð

whatt

ľ³æ (ÕýʽдÊÖ)

¡¾´ð°¸¡¿Ó¦Öú»ØÌû

¡ï
¸Ðл²ÎÓ룬ӦÖúÖ¸Êý +1
mollyzhang: ½ð±Ò+1, ¡ïÓаïÖú 2013-11-11 15:39:22
ÄãÒÔʲô¹Ø¼ü´Ê¼ìË÷µÄ£¿

[ ·¢×ÔСľ³æ¿Í»§¶Ë ]
ÐÄÓжà´ó£¬Ìì¿Õ¾ÍÓжà´ó£¡£¡
2Â¥2013-11-10 22:04:54
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

williamxiang

ľ³æ (ÖøÃûдÊÖ)


¡¾´ð°¸¡¿Ó¦Öú»ØÌû

¡ï ¡ï ¡ï ¡ï ¡ï
¸Ðл²ÎÓ룬ӦÖúÖ¸Êý +1
mollyzhang: ½ð±Ò+5, ¡ï¡ï¡ïºÜÓаïÖú, лл£¬Çë¶à¶àÖ¸½Ì 2013-11-11 15:39:39
Ç×£¬Äã˵µÄÊÇ×÷ÓÃÓڰеãµÄ»¯ºÏÎﻹÊǰе㵰°×±¾Éí°¡£¿
Èç¹ûÊǰе㱾ÉíµÄ»°£¬
ÎÒ¾õµÃ£º
µÚÒ»£¬×÷ΪһÖÖÓÚÈËÌåÄÚÌìÈ»´æÔÚµÄÎïÖÊ£¬GPR120ÊÇ·ñÊôÓÚרÀû·¨ÒâÒåÉϵĿÍÌåÖµµÃ¿¼ÂÇ¡£¡¶×¨Àû·¨¡·£¨2008Äê°æ£©µÚ25Ìõ¹æ¶¨Á˼¸ÖÖ²»ÊÚÓèרÀûȨµÄ¼¸ÖÖ¿ÍÌ壬GPR120ÓëµÚÒ»¿î¡°¿ÆÑ§·¢ÏÖ¡±ÆÄΪÏàËÆ¡£
µÚ¶þ£¬ÔÚPUBMEDÖмì³ö±¨µÀÓÐGPR120×îÔçµÄÎÄÏ×ÊÇ2003ÄêµÄ£¬×÷Õßµ¥Î»ÊÇDepartment of Neuroscience, Uppsala University, BMC¡­¡­Òò´Ë£¬ÕâÒ»µ°°×ÖÁÉÙÔÚ2003Äê»ò¸üÔç¼´ÒѽøÈ빫֪ÁìÓò£¬ËùÒÔ¼´Ê¹Äã˵µÄÄÇЩ¹«Ë¾±Ü¿ª¿ÍÌåÉó²éÕϰ­¶øÏò¸÷רÀû¾ÖµÝ½»ÉêÇ룬Ҳ»áÒòΪ²»´æÔÚÐÂÓ±ÐÔ¶ø±»²µ»Ø¡£Ò»°ãµÄ¹«Ë¾ÊDz»»á×öÕâÖÖ´Àʵġ£
3Â¥2013-11-11 08:40:49
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû

mollyzhang

Ìú¸Ëľ³æ (ÖøÃûдÊÖ)

ÒýÓûØÌû:
2Â¥: Originally posted by whatt at 2013-11-10 22:04:54
ÄãÒÔʲô¹Ø¼ü´Ê¼ìË÷µÄ£¿

ÎÒÊÇÒòΪÔÚÌÀÄ·Ñ·Öв鵽ÒÔÉϵĹ«Ë¾ÔÚ×ö¸Ã°Ðµã, ËùÒÔÊÇÒÔ¹«Ë¾Ãû³Æ¼ìË÷µÄ,Æä´ÎÎÒÒÔ GPR120 (FFA4)Ò²¶¼Ã»ËÑË÷µ½ÉÏÊö¹«Ë¾µÄרÀû
4Â¥2013-11-11 15:37:04
ÒÑÔÄ   »Ø¸´´ËÂ¥   ¹Ø×¢TA ¸øTA·¢ÏûÏ¢ ËÍTAºì»¨ TAµÄ»ØÌû
×î¾ßÈËÆøÈÈÌûÍÆ¼ö [²é¿´È«²¿] ×÷Õß »Ø/¿´ ×îºó·¢±í
[¿¼ÑÐ] »¯¹¤Çóµ÷¼Á£¡ +17 RichLi_ 2026-04-06 17/850 2026-04-06 22:26 by qlm5820
[¿¼ÑÐ] µ÷¼Á +3 mcbbc 2026-04-06 4/200 2026-04-06 20:58 by lbsjt
[¿¼ÑÐ] 315Çóµ÷¼Á +5 £¦123456789 2026-04-05 5/250 2026-04-05 19:55 by nepu_uu
[¿¼ÑÐ] 288Çóµ÷¼Á£¬Ò»Ö¾Ô¸»ªÄÏÀí¹¤´óѧ071005 +6 ioodiiij 2026-04-04 6/300 2026-04-05 10:09 by guoweigw
[¿¼ÑÐ] 353Çóµ÷¼Á +10 MayUxw1 2026-04-03 10/500 2026-04-05 09:23 by Î޼ʵIJÝÔ­
[¿¼ÑÐ] 085602µ÷¼Á ³õÊÔ×Ü·Ö335 +12 19123253302 2026-04-04 12/600 2026-04-05 08:08 by 544594351
[¿¼ÑÐ] ²ÄÁÏר˶322·Ö +11 ¹þ¹þ¹þºðºðºð¹þ 2026-04-02 11/550 2026-04-04 23:37 by ÓÀ×ÖºÅ
[¿¼ÑÐ] 294Çóµ÷¼Á +6 Grey_Ey 2026-04-02 9/450 2026-04-04 22:07 by hemengdong
[¿¼ÑÐ] Ò»Ö¾Ô¸»¦9£¬ÇóÉúÎïѧµ÷¼Á£¬326·Ö +6 Áõīī 2026-04-04 6/300 2026-04-04 19:44 by ÌÆãå¶ù
[¿¼ÑÐ] 359Çóµ÷¼Á +7 hhhhaaaa$ 2026-04-04 7/350 2026-04-04 18:49 by imissbao
[¿¼ÑÐ] 22408Çóµ÷¼Á 354·Ö ¿É¿çרҵ +3 hannnnnnn 2026-04-04 3/150 2026-04-04 14:35 by ÍÁľ˶ʿÕÐÉú
[¿¼ÑÐ] ±¾¿Æ211£¬×¨Òµ085404£¬293·ÖÇëÇóµ÷¼Á +5 Á«²Ë¾ÍÊÇź°É 2026-04-04 5/250 2026-04-04 14:08 by ÕâÊÇÒ»¸öÎÞÁĵÄê
[¿¼ÑÐ] ¿¼Ñе÷¼Á +4 zybz³å³å³å 2026-04-03 6/300 2026-04-04 13:08 by zybz³å³å³å
[¿¼ÑÐ] 294Çóµ÷¼Á +6 Grey_Ey 2026-04-03 6/300 2026-04-03 20:46 by ÐÀϲ777
[¿¼ÑÐ] 372·Ö²ÄÁÏÓ뻯¹¤£¨085600£©Ò»Ö¾Ô¸ºþÄÏ´óѧÇóµ÷¼Á +3 À¶¼ãƬ 2026-04-03 4/200 2026-04-03 17:58 by Jimmyandyou
[¿¼ÑÐ] Çóµ÷¼Á +7 Aniyaio 2026-04-02 7/350 2026-04-02 16:42 by zzsw+
[¿¼ÑÐ] 285Çóµ÷¼Á +11 AZMK 2026-04-01 11/550 2026-04-01 22:40 by peike
[¿¼ÑÐ] 286Çóµ÷¼Á +5 Sa67890. 2026-04-01 7/350 2026-04-01 19:50 by 6781022
[¿¼ÑÐ] 353Çóµ÷¼Á +4 À­¹³²»Ðí±ä 2026-04-01 4/200 2026-04-01 18:10 by ¼Çʱ¾2026
[˶²©¼ÒÔ°] ²©Ò»±»ËͳöÁªÅà¸Ð¾õ²»ÊÊÓ¦Ôõô°ì +3 È«´åµÄ¹· 2026-03-31 3/150 2026-04-01 10:44 by 328838485
ÐÅÏ¢Ìáʾ
ÇëÌî´¦ÀíÒâ¼û