| ²é¿´: 964 | »Ø¸´: 11 | |||
| µ±Ç°Ö÷ÌâÒѾ´æµµ¡£ | |||
yanhongsenľ³æ (ÕýʽдÊÖ)
|
[½»Á÷]
ÖÐÒ©³É·ÖµÄÎüÊÕ¡¢·Ö²¼¡¢´úл¡¢ÅÅй¡¢¶¾ÐÔÓëҩЧ
|
||
|
¡¾ÄÚÈݽéÉÜ¡¿ ±¾Êé×ܽáÁËÖÐÒ©³É·ÖµÄÎüÊÕ¡¢·Ö²¼¡¢´úл¡¢ÅÅйºÍ¶¾ÐÔ(ADME£¯Tox£®) ÒÔ¼°Ïà¹ØÒ©Ð§µÄÑо¿³É¹û£¬È«Êé·ÖÉÏ¡¢ÏÂÁ½Æª¡£ÉÏÆªÎª×ÜÂÛ£»ÏÂÆªÎª¸÷ÂÛ£¬ ·Ö°ËÕ£¬°´ÖÐÒ©»¯Ñ§³É·Ö½á¹¹ÀàÐÍ·ÖÀ࣬ÊÕÔØÖÐÒ©³É·Ö475¸ö£¬È«Êé280ÓàÍò ×Ö¡£Ã¿¸öÖÐÒ©»¯Ñ§³É·ÖÌõÄ¿°üÀ¨£º¡¾»¯Ñ§Ãû¡¿¡¢¡¾Ó¢ÎÄÃû¡¿¡¢¡¾ÒìÃû¡¿¡¢¡¾ ½á¹¹Ê½¡¿¡¢¡¾·Ö×Óʽ¼°·Ö×ÓÁ¿¡¿¡¢¡¾À´Ô´¡¿¡¢¡¾ADME£¯Tox£®¡¿¡¢¡¾ÉúÎï»î ÐÔ¡¿¡¢¡¾·ÖÎö·½·¨¡¿¡¢¡¾»¯Ñ§½á¹¹Æ×ѧÊý¾Ý¡¿¡¢¡¾¸½¼Ç¡¿ºÍ¡¾²Î¿¼ÎÄÏס¿µÈ Ê®¶þ¸ö²¿·Ö¡£ÄÚÈݷḻ¡¢ÎÄͼÏèʵ¡¢¿ÆÑ§ÐÔÇ¿£¬¿É¹©»îÔ¾ÔÚÖÐÒ©ÏÖ´ú»¯Ñо¿ µÄ¿ÆÑй¤×÷Õߺ͹ã´óÖÐÒ½Ò©¼°ÖÐÎ÷Ò½½áºÏ¹¤×÷ÕßÒÔ¼°Ïà¹ØË¶Ê¿¡¢²©Ê¿Ñо¿Éú ²Î¿¼¡£ ¡¾±¾ÊéĿ¼¡¿ ÉÏÆª ×ÜÂÛ µÚÒ»Õ Ð÷ÂÛ µÚ¶þÕ ÌåÄÚÒ©ÎïŨ¶È·¨ µÚÈýÕ ÉúÎïЧӦ·¨ µÚËÄÕ ҩÎïѧºÍҩЧѧ½áºÏÄ£ÐÍ µÚÎåÕ ÖÐÒ©Ò©¶¯Á¦Ñ§µÄÐÂѧ˵ºÍз½·¨ µÚÁùÕ ÖÐÒ©Ò©´ú¶¯Á¦Ñ§µÄÄѵ㡢ÈȵãºÍ¶Ô²ß ÏÂÆª ¸÷ÂÛ µÚÒ»Õ ֬·¾×廯ºÏÎï µÚ¶þÕ ·¼Ïã×廯ºÏÎï µÚÈýÕ Ñõ»¯ÔÓ»·»¯ºÏÎï µÚËÄÕ ֬»·×廯ºÏÎï µÚÎåÕ ÉúÎï¼î µÚÁùÕ ¿óÎïÀàÖÐÒ©³É·Ö µÚÆßÕ µ°°×ÀàÖÐÒ©³É·Ö µÚ°ËÕ ÌÇÀàÖÐÒ©³É·Ö Ë÷Òý ¸½Â¼ ADME/Tox./Act.Ñо¿Öеij£ÓÃÊõÓï ¸öÈ˾õµÃÕâ±¾ÊéºÜºÃµÄ£¬ËÓÐûÓеç×Ó°æµÄ°¡ ¹²Ïíһϣ¬½è´Ë·¢¶¯Ò©³æÒ»ÆðѰÕÒһϣ¬¹ºÂòÌ«¹óÁËЩ°¡ |
» ²ÂÄãϲ»¶
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ8È˻ظ´
ÌåÖÆÄÚ³¤±²ËµÌåÖÆÄÚ¾ø´ó²¿·ÖÒ»±²×ÓÔڵײ㣬ÈçͬÄãÃÇÒ»Ñù´ó²¿·ÖÆÕͨ½ÌʦæÇÒÊÕÈëµÍ
ÒѾÓÐ13È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ8È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ8È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ11È˻ظ´
ΪʲôÖйú´óѧ¹¤¿Æ½ÌÊÚÃÇË®ÁËÄÇô¶àËùνµÄ¶¥»á¶¥¿¯£¬µ«»¹ÊÇ×ö²»³öÓîÊ÷»úÆ÷ÈË£¿
ÒѾÓÐ8È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ5È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ6È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ9È˻ظ´
ÊÛSCIÒ»ÇøÎÄÕ£¬ÎÒ:8 O5 51O 54,¿ÆÄ¿ÆëÈ«,¿É+¼±
ÒѾÓÐ4È˻ظ´
» ±¾Ö÷ÌâÏà¹ØÉ̼ÒÍÆ¼ö: (ÎÒÒ²ÒªÔÚÕâÀïÍÆ¹ã)
boss126
Òø³æ (СÓÐÃûÆø)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 499
- Ìû×Ó: 84
- ÔÚÏß:
- ³æºÅ: 99705
- ×¢²á: 2005-11-11
- ÐÔ±ð: GG
2Â¥2007-11-27 12:25:59
yanhongsen
ľ³æ (ÕýʽдÊÖ)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 2422.1
- ºì»¨: 2
- Ìû×Ó: 444
- ÔÚÏß: 82.1Сʱ
- ³æºÅ: 230024
- ×¢²á: 2006-03-26
- ÐÔ±ð: GG
- רҵ: ͨÐÅÀíÂÛÓëϵͳ
3Â¥2007-11-27 17:27:36
marshalking
ͳæ (СÓÐÃûÆø)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 117.8
- Ìû×Ó: 122
- ÔÚÏß: 6.7Сʱ
- ³æºÅ: 441585
- ×¢²á: 2007-10-27
- ÐÔ±ð: GG
- רҵ: ÖÐÒ©»¯Ñ§
4Â¥2007-12-03 22:48:55
marshalking
ͳæ (СÓÐÃûÆø)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 117.8
- Ìû×Ó: 122
- ÔÚÏß: 6.7Сʱ
- ³æºÅ: 441585
- ×¢²á: 2007-10-27
- ÐÔ±ð: GG
- רҵ: ÖÐÒ©»¯Ñ§
5Â¥2007-12-03 22:52:46
6Â¥2007-12-06 07:52:38
yjhorn
ľ³æ (ÕýʽдÊÖ)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 1725.8
- Ìû×Ó: 629
- ÔÚÏß: 18.3Сʱ
- ³æºÅ: 33078
- ×¢²á: 2003-12-28
- ÐÔ±ð: GG
- רҵ: ½ðÈÚѧ

7Â¥2007-12-06 08:54:15
flywilling
ͳæ (³õÈëÎÄ̳)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 194.5
- Ìû×Ó: 26
- ÔÚÏß: 51·ÖÖÓ
- ³æºÅ: 448904
- ×¢²á: 2007-11-02
- ÐÔ±ð: MM
- רҵ: ΢ÉúÎïÓëÉú»¯Ò©Ñ§
8Â¥2007-12-06 08:59:33
yanhongsen
ľ³æ (ÕýʽдÊÖ)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 2422.1
- ºì»¨: 2
- Ìû×Ó: 444
- ÔÚÏß: 82.1Сʱ
- ³æºÅ: 230024
- ×¢²á: 2006-03-26
- ÐÔ±ð: GG
- רҵ: ͨÐÅÀíÂÛÓëϵͳ
9Â¥2007-12-07 08:55:57
zhangknme
ľ³æ (СÓÐÃûÆø)
- Ó¦Öú: 0 (Ó×¶ùÔ°)
- ½ð±Ò: 3188.4
- Ìû×Ó: 172
- ÔÚÏß: 15Сʱ
- ³æºÅ: 92482
- ×¢²á: 2005-09-09
- רҵ: Ò©ÎïѧÆäËû¿ÆÑ§ÎÊÌâ

10Â¥2007-12-07 10:22:20













»Ø¸´´ËÂ¥
