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yin198716

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In addition, DLL4-blocking agents have been shown to lack the adverse effect of goblet cell metaplasia, which is a dose-limiting factor for GSIs. Thus, DLL4 inhibitors appeared to be a promising agent for cancer therapy. However, it has been shown that chronic Dll4 inhibition can cause pathological activation of endothelial cells and consequently vascular neoplasms.
Oncology
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andrewzhang

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yin198716: 金币+5, 翻译EPI+1 2013-08-03 00:47:01
此外,DLL4阻断剂已经被证明对于杯状细胞的异变没有负面影响(GSIs对于杯状细胞的影响是其使用剂量受限的重要原因)。因此,DLL4抑制剂今后在癌症治疗中的使用看起来前途光明。然而,也有研究表明,DLL4会导致内皮细胞的病理性激活从而可能引发血管瘤。
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