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We introduced morpholine to form hydrogen bonds with Glu-61 in the c-subunit of ATP synthase and prevent proton transport which is necessary for the synthesis of ATP .£¨¼ÓЩʲôʹÆäÁ¬¹áÄØÕâÀWe introduced adamantine to get better lipophilicity and selectivity.

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baiyuefei(½ð±Ò+15, ·­ÒëEPI+1): 2011-06-27 17:17:04
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We introduced morpholine to form hydrogen bonds with Glu-61 in the c-subunit of ATP synthesis and prevent proton transport. However, the proton transport is a necessary (and important) step in the synthesis of ATP. Therefore, we introduced adamantine to get better lipophilicity and selectivity.
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baiyuefei(½ð±Ò+5): 2011-06-27 17:17:11
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... Therefore, adamantine is incorporated to get better lipophilicity and selectivity.
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