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some compounds inhibit the activity of multidrug efflux transporters responsible for multixenobiotic resistance (MXR) in gills of marine mussels at low exposure levels


Further, weak estrogenic effects were observed at relatively high concentrations
and antiestrogenic activities were found in various cell lines even at very low concentrations, thus showing these compounds to be selective estrogen receptor modulators (SERMs), inducing both estrogenic and antiestrogenic activity, dependent on cell line and ER subtype targeted (Schreurs et al., 2002).

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