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Literature References:  DNA topoisomerase I inhibitor.  Semisynthetic derivative of camptothecin, q.v.; de-esterified in vivo to the active metabolite, 7-ethyl-10-hydroxycamptothecin (SN-38).  Prepn:  JP Kokai 85 19790; T. Miyasaka et al., US 4604463 (1985, 1986 both to Yakult Honsha); S. Sawada et al., Chem. Pharm. Bull. 39, 1446 (1991).  Antitumor activity and toxicity data:  T. Kunimoto et al., Cancer Res. 47, 5944 (1987).  Mechanism of action study:  Y. Kawato et al., ibid. 51, 4187 (1991).  Clinical trial in colorectal cancer:  J. Y. Douillard et al., Lancet 355, 1041 (2000).  Review of pharmacology and clinical experience:  N. Masuda et al., Crit. Rev. Oncol. Hematol. 24, 3-26 (1996); S. O'Reilly, E. K. Rowinsky, ibid. 47-70.
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