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ÇóÖú´óÉñ°ïÎÒÏÂÔØÒ»ÆªÍâÎĵÄÎÄÏ×£¬Ð»Ð»£¡ Title: Discovery of 1-{4-[1-(2,6-Difluorobenzyl)-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl]phenyl}-3-methoxyurea (TAK-385) as a Potent, Orally Active, Non-Peptide Antagonist of the Human Gonadotropin-Releasing Hormone Receptor Source: Journal of Medicinal Chemistry (formerly: Journal of Medicinal and Pharmaceutical Chemistry) [0022-2623] Miwa yr:2011 vol:54 iss:14 pg:4998 -5012 |
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