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Q邱邱

新虫 (小有名气)

[求助] 求克罗烷药理作用及研究意义

在线等,挺急的,重金悬赏,哈哈哈

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mac194

铁虫 (职业作家)

【答案】应助回帖

研究意义:

  http://grantome.com/grant/NIH/R01-GM039075-03  "Total Synthesis of Clerodane Diterpenes"

Clerodanes are a group of diterpenoid natural products which have been found to possess a broad spectrum of biological activity. Some have been shown to be potent insect antifeedants. Others have been found to have antitumor, antimicrobial, antifungal, antiviral, or antiulcer activity **...

**1998... 新发现益处更值得关注


药理作用:

  我实在外行, 只能建议你看这篇国内教授写的综论文章

    pubs.rsc.org/en/content/articlelanding/2016/np/c5np00137d
2楼2018-06-04 06:52:22
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Q邱邱

新虫 (小有名气)

引用回帖:
2楼: Originally posted by mac194 at 2018-06-04 06:52:22
研究意义:

  http://grantome.com/grant/NIH/R01-GM039075-03  "Total Synthesis of Clerodane Diterpenes"

Clerodanes are a group of diterpenoid natural products which have been fo ...

研究意义……意义……意义……不是呀

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3楼2018-06-04 14:41:32
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mac194

铁虫 (职业作家)

引用回帖:
3楼: Originally posted by Q邱邱 at 2018-06-04 14:41:32
研究意义……意义……意义……不是呀
...

意义是:

  可同时施展多种奇特药效 (抗良性瘤/恶性癌, 对付耐药性, 减轻阿片依赖 的单个分子不多

  血脑屏障很难很难绕过 (2016 后才真有进步*), 精准定时释放药物的科技麻省理工学院去年底才刚公布**

  有鉴于此, 大部分公私构选择赞助 药性浅缓/临床试验简单 的天然产品研究

  * http://news.cornell.edu/stories/ ... in-diseases-cancers

    https://vector.childrenshospital ... lood-brain-barrier/


** http://www.sohu.com/a/208055202_100074008
4楼2018-06-04 20:24:52
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