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Pentacyclic triterpenoids  which have a wide range of biological activity  is a class of widely exist in nature,and the anti-tumor effect is one of its main activities. It works in  inhibiting tumor cell proliferation and angiogenesis, inducing tumor cell apoptosis and reversaling of drug resistance. As its complex and diverse mechanism which contains several targets,the pentacyclic triterpenoids has become a lead class of potential anti-tumor compounds and caused  global extencive attention on the  field of antineoplastic drugs. The paper reviews
the mechanism of anti-tumor research in recent years.
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