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ÎÊÌâ1£º¡°All of the mass spectra reported in this work are very difficult to read. The quality of these spectra needs to be enhanced. Why are the signal levels in the mass spectra lower than that typically seen in MS characterization of organic compounds(1e5 to 1e6). Please provide total ion chromatogram (TIC) for all the compounds for which the 1-H NMR has been provided. ¡°
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ÎÊÌâ2£º¡±        In the section on X-ray crystallography, why did dichlormethane take 7days to evaporate at room temperature?  Also the R values for refinement of the crystal structure (0.07) is too high. Typically the R factor should be less than 3%. ¡°
µ±Ê±ÓÃÁËDCMÑøµ¥¾§£¬ËµÊµ»°ÎÒÒ²²»¼ÇµÃÊǶà¾Ã²ÅÎö³öµ¥»úµÄ£¬Ö»ÊǹýÁËÒ»¸öÀñ°Ý£¬È¥¿´ÁËÏ£¬Óе¥¾§ÁË£¬ÎÒ¾ÍÏ¡ÀïºýÍ¿µÄдÁË7ÌìÎö³öµ¥¾§£¬ÏÖÔÚÏëÏëȷʵ²»ºÏ³£Àí£»Éó¸åÈËÒ²Ìáµ½ÎÒRÖµµÄÎÊÌ⣬µ¥¾§ÎÒÒ²²»ÊÇÌ«¶®£¬ºÃÏñûÓÐÕÒµ½ÎÒµÄRÖµ£¬²»ÖªµÀ²»»Ø´ð»á²»»áÓÐÎÊÌâ

ÎÊÌâ3£º¡±The manuscript should be completed for e.g. logP, logS, pKa, PSA data and SAR relations of compounds studied discussed in more quantitative way.¡°
СµÜÎÒÕæÐIJ»ÖªµÀ¡±logP, logS, pKa, PSA data and SAR relations of compounds¡°ÎªºÎÎ²»ÖªµÀÊDzâ³öÀ´µÄ»¹ÊǼÆËã³öÀ´µÄ£¬»¹Çë¸÷λ´óÏÀ¶à¶àÖ¸½Ì£¡

[ Last edited by ·¨¹Ùliu on 2014-8-25 at 11:02 ]
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35Â¥: Originally posted by jeangong at 2014-08-25 11:57:53
logP£ºpartition-coefficient ·ÖÅäϵÊý£ºÎïÖÊÔÚ֬ˮÁ½ÏàÖзÖÅäϵÊýµÄ¶ÔÊýÖµ£¬Óл¯ºÏÎïÊèË®³£ÊýClogPºÍ·Ö×ÓÊèË®³£ÊýMlogP»¯ºÏÎïµÄ²ÎÊý£¬¼ÆËã³öÀ´µÄ,

logS, ÎÒ²»ÖªµÀ£¬Ó¦¸ÃºÍlogP²î²»¶à£¬ÎïÖʵÄÐÔÖʵÄÒ»ÖÖ²ÎÊý£¬¿É ...

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